Fluorine in pharmaceutical industry: fluorine-containing drugs introduced to the market in the last decade (2001-2011).

Keywords

Library science, China, Political science, Humanities, Art

References

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• A trifluorinated thiazoline scaffold leading to pro-apoptotic agents targeting prohibitins.由子 稲垣 — 2014
• Palladium(II)-catalyzed directed trifluoromethylthiolation of unactivated C(sp³)-H bonds.Patricia Andrés González — 2015
• Benzylic C(sp(3) )H Perfluoroalkylation of Six-Membered Heteroaromatic Compounds.Éric Perron — 2015
• Photoredox-Catalyzed Tandem Insertion/Cyclization Reactions of Difluoromethyl and 1,1-Difluoroalkyl Radicals with Biphenyl Isocyanides.R. J. Braddock, R.A. Dennison, E.M. Ahmed — 2015
• Pentafluorosulfanyl-containing flufenamic acid analogs: Syntheses, properties and biological activities勝次 山野 — 2015
• New Diethyl Ammonium Salt of Thiobarbituric Acid Derivative: Synthesis, Molecular Structure Investigations and Docking StudiesAaron H. Groth, Paul Mirski, T. Zangerl — 2015
• (18)F-Labeling of Arenes and Heteroarenes for Applications in Positron Emission Tomography.José Benedito Alberola — 2016
• Microsolvation of Fluoromethane.van W.M.J. Kessel — 2016
• A redox-economical synthesis of trifluoromethylated enamides with the Langlois reagent.Sri Sumarsih, Dr.Ir. Y. Marsono — 2017
• Activation of SF6 at Platinum Complexes: Formation of SF3 Derivatives and Their Application in Deoxyfluorination Reactions.María Bauluz del Río, Soledad Arias Senso, Andrés López de Alda González — 2017
• Cu-Catalyzed Aminodifluoroalkylation of Alkynes and α-Bromodifluoroacetamides.Patricia Pérez Zaragoza, Oscar Torres Pereira — 2017
• Synthesis of 4-(Trifluoromethyl)cyclopentenones and 2-(Trifluoromethyl)furans by Reductive Trifluoroacetylation of Ynones.J. G. Phillips, E. Hernández Balada, William N. Marmer — 2017
• Iron-catalyzed ortho trifluoromethylation of anilines via picolinamide assisted photoinduced C-H functionalization.François Coussens — 2018
• Pd(II)-Catalyzed Carbonyl-Directing Activation of Alkenes: Selective Fluorosulfonylation and Aminosulfonylation of 1,7-Enynes.Barbara Hallensleben — 2018
• Ligand-Based Fluorine NMR Screening: Principles and Applications in Drug Discovery Projects.John D. Gearhart — 2018
• Leaving Group Assisted Strategy for Photoinduced Fluoroalkylations Using N-Hydroxybenzimidoyl Chloride Esters.Ivonnet Arcia Zamora — 2018
• Perfluorophenyl Derivatives as Unsymmetrical Linkers for Solid Phase ConjugationPatricia Y. Hashima — 2018
• eToxPred: a machine learning-based approach to estimate the toxicity of drug candidatesJosé Antonio Fernández Ordóñez — 2019
• Shelf-stable electrophilic reagents for trifluoromethylthiolation.Xinxin Shao, Chunfa Xu, Long Lü — 2015
• Substrate stereocontrol in bromine-induced intermolecular cyclization: asymmetric synthesis of pitavastatin calciumWeiqi Chen, Fangjun Xiong, Qian Liu — 2015

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