Pharmacology of cannabinoid CB1 and CB2 receptors.
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Summary
This review focuses on the classification, binding properties, effector systems and distribution of cannabinoid receptors, and describes the various cannabinoid receptor agonists and antagonists now available and considers the main in vivo and in vitro bioassay methods that are generally used.
- Type
- review
- Published
- 1997-01-01
- Cited by
- 1,514
- References
- 183
- OpenAlex
- https://openalex.org/W2015614945
- Semantic Scholar
- https://api.semanticscholar.org/CorpusID:46569473
Keywords
Cannabinoid receptor, Cannabinoid, GPR18, Receptor, Cannabinoid receptor type 2
References
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Cited by
- Changes in the Endocannabinoid system in the Brain Following Bilateral Vestibular Damage
- EDG6, a novel G-protein-coupled receptor related to receptors for bioactive lysophospholipids, is specifically expressed in lymphoid tissue.
- D2 dopamine receptors enable Δ9‐tetrahydrocannabinol induced memory impairment and reduction of hippocampal extracellular acetylcholine concentration
- Cannabinoid receptor agonists inhibit depolarization‐induced calcium influx in cerebellar granule neurons
- Coexpression of the cannabinoid receptor type 1 with dopamine and serotonin receptors in distinct neuronal subpopulations of the adult mouse forebrain.
- Anandamide‐induced neuroblastoma cell rounding via the CB1 cannabinoid receptors
- Functions of cannabinoid receptors in the hippocampus.
- Tetrahydrocannabinol and endocannabinoids in feeding and appetite.
- Binding of anandamide to bovine serum albumin Published, JLR Papers in Press, July 1, 2003. DOI 10.1194/jlr.M300170-JLR200
- Marijuana and cannabinoid regulation of brain reward circuits
- Synthesis and SAR of 5,6-diarylpyridines as human CB1 inverse agonists.
- Evaluation of the in vivo receptor occupancy for the behavioral effects of cannabinoids using a radiolabeled cannabinoid receptor agonist, R‐[125/131I]AM2233
- Cannabinoids enhance susceptibility of immature brain to ethanol neurotoxicity
- Design and Synthesis of (13S)-Methyl-Substituted Arachidonic Acid Analogues: Templates for Novel Endocannabinoids
- Cannabinoid receptor signaling.
- Decreased frontal N-acetylaspartate levels in adolescents concurrently using both methamphetamine and marijuana
- Effects of cannabinoids and related fatty acids upon the viability of P19 embryonal carcinoma cells
- Structural requirements for cannabinoid receptor probes.
- Discovery of a high affinity and selective pyridine analog as a potential positron emission tomography imaging agent for cannabinoid type 2 receptor.
- Pharmacological characterization of rat VD-hemopressin(α), an α-hemoglobin-derived peptide exhibiting cannabinoid agonist-like effects in mice.
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