Mechanisms for activation and antagonism of an AMPA-sensitive glutamate receptor: crystal structures of the GluR2 ligand binding core.

Keywords

AMPA receptor, Kainate receptor, DNQX, Chemistry, Allosteric regulation

References

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Cited by

• Chemical scale investigations of ligand-gated ion channels using unnatural amino acidsDarren L. Beene — 2005
• Universality of receptor channel responses.Listi Erawaty Simbolon — 2001
• Differential activation of individual subunits in heteromeric kainate receptors.José Luis Pablos Rodríguez, Mónica Álvarez — 2002
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• Glutamate receptor ion channels: where do all the calories go?James P. Kauahikaua, Charles J. Zablocki, Dallas B. Jackson — 2011
• Structural Mechanism of N-Methyl-D-Aspartate Receptor Type 1 Partial AgonismSandra D. Pearce — 2012
• CrossTalk proposal: TARPs modulate AMPA receptor gating transitionsРоманова Татьяна Владимировна — 2013
• Understanding The Single Channel Behavior Of Glua3 ReceptorsKinning Poon — 2011
• Handbook of ion channelsJie Zheng, M. Trudeau — 2015
• Structure/function studies of the P2X receptorHelen Digby — 2007
• Positions in the glun2c-containing nmdar regulate alcohol sensitivity and ion channel gatingMan Wu — 2014
• Spectroscopic and kinetic methods for ligand-protein interactions of glutamate receptor.Vasanthi Jayaraman — 2004
• Extracellular Modulation of NMDA ReceptorsKeith Williams — 2009
• A Spatial Model of the Glycine Site of the NR1 Subunit of NMDA-Receptor and Ligand DockingIrina G. Tikhonova, Igor I. Baskin, Vladimir A. Palyulin — 2004
• Synaptic plasticity regulated by protein-protein interactions and posttranslational modifications.Norihiko Yokoi, Masaki Fukata, Yuko Fukata — 2012
• Computational Approaches in Molecular and Systems Pharmacology: Application to Neurosignaling Membrane ProteinsChang Liu — 2014
• Regulation of calcium-permeable AMPA receptors in gliaM. Zonouzi — 2011
• Molecular Modeling of the Ligand-Binding Domains of the NR3A and NR3B Subunits of the NMDA ReceptorBelenikin Ms, Gabriele Costantino, Vladimir A. Palyulin — 2003

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