X-Ray Structures and Analysis of 11 Cyclosporin Derivatives Complexed with Cyclophilin A.

Keywords

Medicine

References

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• X-ray structure of alisporivir in complex with cyclophilin A at 1.5 Å resolution.Alexa Diéguez — 2018
• Using Molecular Dynamics to Elucidate the Mechanism of CyclophilinLauren McGowan — 2014
• Probing protein-ligand interactions via solution phase hydrogen exchange mass spectrometryStefan T. Esswein — 2010
• Effects of ligand binding on the rigidity and mobility of proteins : a computational and experimental approachJack W. Heal — 2013
• Two structures of cyclophilin 40: folding and fidelity in the TPR domains.Paul Taylor, Jacqueline Dornan, Amerigo Carrello — 2001
• Synthesis and characterization of constrained cyclosporin A derivatives containing a pseudo-proline groupLuc Patiny, Jean‐François Guichou, Michael Keller — 2003
• Exo‐Mechanism Proximity‐Accelerated Alkylations: Investigations of Linkers, Electrophiles and Surface Mutations in Engineered Cyclophilin–Cyclosporin SystemsKonstantín L. Levitsky, Melissa Boersma, Christopher J. Ciolli — 2005
• Two new cyclosporin folds observed in the structures of the immunosuppressant cyclosporin G and the formyl peptide receptor antagonist cyclosporin H at ultra-high resolution.B.S. Potter, Rex A. Palmer, Robert Withnall — 2003
• Immunophilins and HIV-1 V3 Loop For Structure-Based Anti-AIDS Drug DesignAlexander M. Andrianov — 2009
• Thermodynamics of the cyclophilin-A/cyclosporin-A interaction: a direct comparison of parameters determined by surface plasmon resonance using Biacore T100 and isothermal titration calorimetry.Martin A. Wear, Malcolm D. Walkinshaw — 2006
• Structure of a bacterial cytoplasmic cyclophilin A in complex with a tetrapeptide.Elias Christoforides, Maria Dimou, Panagiotis Katinakis — 2012
• Equilibrium unfolding of cyclophilin from Leishmania donovani: characterization of intermediate states.Sourav Roy, Sankar Basu, Alok K. Datta — 2014
• Immunophilins: Switched on protein binding domains?Michael T. G. Ivery — 2000
• 1.88 A crystal structure of the C domain of hCyP33: a novel domain of peptidyl-prolyl cis-trans isomerase.Tao Wang, Cai‐Hong Yun, Shenyan Gu — 2005
• Computational Model of the HIV-1 Subtype A V3 Loop: Study on the Conformational Mobility for Structure-Based Anti-AIDS Drug DesignAlexander M. Andrianov, Ivan Anishchenko — 2009
• The three-dimensional structure of a Plasmodium falciparum cyclophilin in complex with the potent anti-malarial cyclosporin A.Mark R. Peterson, David R. Hall, Matthew Berriman — 2000
• Structural and Biochemical Characterization of the Human Cyclophilin Family of Peptidyl-Prolyl IsomerasesTara L. Davis, John R. Walker, Valérie Campágna‐Slater — 2010
• Preparation, Characterization and Refolding in Vitro of a Recombinant Human Cyclophilin A Mutant: Effect of a Single Pro/Ser Substitution on Cyclophilin A Structure and PropertiesLi‐Ren Xu, Xiao Yan, Man Luo — 2008
• Structural basis for the non-immunosuppressive character of the cyclosporin A analogue Debio 025.Isabelle Landrieu, Xavier Hanoulle, Fanny Bonachéra — 2010
• Enzymatic and structural characterization of non-peptide ligand-cyclophilin complexes.George Kontopidis, Paul Taylor, Malcolm D. Walkinshaw — 2004

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