Pd-Catalyzed C-H aziridination of 3,3,5,5-tetrasubstituted piperazin-2-ones.
Explore this paper's citation graph
Summary
A palladium mediated C-H aziridination reaction of 3,3,5,5-substituted-piperazin-2-ones has been developed using phenyliodonium diacetate (PIDA) and succinic acid to give synthetically useful bicyclic Aziridines, in moderate to good yields.
- Type
- article
- Published
- 2017-12-04
- Cited by
- 4
- References
- 27
- OpenAlex
- https://openalex.org/W2771393740
- Semantic Scholar
- https://api.semanticscholar.org/CorpusID:46281645
Keywords
Chemistry, Catalysis, Combinatorial chemistry, Medicinal chemistry, Stereochemistry
References
- Ligand-Enabled Catalytic C-H Arylation of Aliphatic Amines by a Four-Membered-Ring Cyclopalladation Pathway.
- Palladium-Catalysed, Directed CH Coupling with Organometallics
- Discovery of N-Aryl Piperazines as Selective mGlu5 Potentiators with Efficacy in a Rodent Model Predictive of Anti-Psychotic Activity
- Challenge and progress: palladium-catalyzed sp3 C–H activation
- TEMPO and Its Derivatives: Synthesis and Applications
- Platinum model studies for palladium-catalyzed oxidative functionalization of C-H bonds
- Lithium 2,2,6,6-tetramethylpiperidide and related, strong, proton-specific bases. Evaluation in synthesis
- Synthetic and Mechanistic Studies of Pd-Catalyzed C–H Arylation with Diaryliodonium Salts: Evidence for a Bimetallic High Oxidation State Pd Intermediate
- Palladium-catalysed C–H activation of aliphatic amines to give strained nitrogen heterocycles
- The First Dinuclear Complex of Palladium(III)
- Synthetically important alkali-metal utility amides: lithium, sodium, and potassium hexamethyldisilazides, diisopropylamides, and tetramethylpiperidides.
- Industrial Oxidations with Organocatalyst TEMPO and Its Derivatives
- Microwave-Assisted Catalyzed Asymmetric Transformations of Natural Products
- Bimetallic Pd(III) complexes in palladium-catalysed carbon–heteroatom bond formation.
- Ring-opening reactions of nonactivated aziridines catalyzed by tris(pentafluorophenyl)borane.
- Serotonin receptor and transporter ligands - current status.
- Controlled Photoradical Polymerization Mediated by 2,2,6,6-Tetramethylpiperidine-1-Oxyl
- High-oxidation-state palladium catalysis: new reactivity for organic synthesis.
- Biologically Active 1-Arylpiperazines. Synthesis of New N-(4-Aryl-1-piperazinyl)alkyl Derivatives of Quinazolidin-4(3H)-one, 2,3-Dihydrophthalazine-1,4-dione and 1,2-Dihydropyridazine-3,6-dione as Potential Serotonin Receptor Ligands
- Off-line coupling of automated pipetting system with square wave voltammetry
Cited by
Related papers
- ФОРМИРОВAНИЕ ГОТОВНОСТИ БУДУЩИХ ПЕДAГОГОВ К ОРГAНИЗAЦИИ РAБОТЫ ПО РAЗВИТИЮ ВAЛЕОЛОГИЧЕСКОЙ КУЛЬТУРЫ ШКОЛЬНИКОВ
- A GEOMETRIC MEAN IN THE FURUTA INEQUALITY
- Darstellung perhalogenierter Dimethyldisulfane durch photochemische Reaktion von CSF2 und CSFCI mit Sulfenylbromiden bzw. ‐chloriden
- Chemistry of the p-block elements with anionic scorpionate ligands
- Chemistry of geminal diazides. Rearrangements to N-Cyano compounds
- Reaktionen mit 3-Chloro-1,2-benzisothiazolium-chloriden. Synthese von 2-substituierten 3-Amino-benzo[b]-thiophenen