The utility of rat jejunal permeability for biopharmaceutics classification system
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Summary
It is concluded that drugs could be categorized correctly based on dose number and their intestinal permeability values in rat model using single-pass intestinal perfusion technique.
- Type
- article
- Published
- 2009-11-20
- Cited by
- 34
- References
- 32
- OpenAlex
- https://openalex.org/W2074668181
- Semantic Scholar
- https://api.semanticscholar.org/CorpusID:207463968
Keywords
Biopharmaceutics Classification System, Intestinal permeability, Jejunum, Permeability (electromagnetism), Biopharmaceutics
References
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- Intestinal Permeability Enhancement: Efficacy, Acute Local Toxicity, and Reversibility
- High in situ rat intestinal permeability of artemisinin unaffected by multiple dosing and with no evidence of P-glycoprotein involvement.
- Molecular properties of WHO essential drugs and provisional biopharmaceutical classification.
- Physicochemical Characterization of Solid Dispersions of Indomethacin with PEG 6000, Myrj 52, Lactose, Sorbitol, Dextrin, and Eudragit® E100
- In vitro systems for studying intestinal drug absorption
- Biopharmaceutic classification system: a scientific framework for pharmacokinetic optimization in drug research.
- Drug, Meal and Formulation Interactions Influencing Drug Absorption After Oral Administration
- LC determination of piroxicam in human plasma.
- The biopharmaceutics classification system (BCS): class III drugs - better candidates for BA/BE waiver?
- Quantitative Biopharmaceutics Classification System: The Central Role of Dose/Solubility Ratio
- Oral absorption of anti-AIDS nucleoside analogues. 1. Intestinal transport of didanosine in rat and rabbit preparations.
- Oral absorption of anti‐ AIDS nucleoside analogues. 3. Regional absorption and in vivo permeability of 2′, 3′ ‐ dideoxyinosine in an intestinal–vascular access port (IVAP) dog model
- Error structure for the HPLC analysis for atenolol, metoprolol and propranolol: a useful weighting method in parameter estimation.
- Use of laminar flow and unstirred layer models to predict intestinal absorption in the rat.
- Biopharmaceutical classification of drugs using intrinsic dissolution rate (IDR) and rat intestinal permeability.
- Characterization of small intestinal transit time distribution in humans
- Transdermal delivery of drugs with differing lipophilicities using azone analogs as dermal penetration enhancers.
Cited by
- Periplocymarin is a potential natural compound for drug development: highly permeable with absence of P‐glycoprotein efflux and cytochrome P450 inhibitions
- Determination of intestinal permeability of rigosertib (ON 01910.Na, Estybon): correlation with systemic exposure
- Systematic development of DoE optimized SNEDDS of sirolimus with enhanced intestinal absorption
- Pharmaceutical Usefulness of Biopharmaceutics Classification System: Overview and New Trend
- Application of Method Suitability for Drug Permeability Classification
- Optimized PLGA nanoparticle platform for orally dosed trans-resveratrol with enhanced bioavailability potential
- An improved prediction of the human in vivo intestinal permeability and BCS class of drugs using the in vitro permeability ratio obtained for rat intestine using an Ussing chamber system
- In Vitro and In Situ Evaluation of pH-Dependence of Atazanavir Intestinal Permeability and Interactions with Acid-Reducing Agents
- Biopharmaceutical classification of drugs using intrinsic dissolution rate (IDR) and rat intestinal permeability.
- A study on enhanced intestinal permeability of clarithromycin nanoparticles
- Hydroxypropyl-sulfobutyl-β-cyclodextrin improves the oral bioavailability of edaravone by modulating drug efflux pump of enterocytes.
- Evidence for Enhanced Intestinal Absorption of Digoxin by P-Glycoprotein Inhibitors
- Design of vancomycin RS-100 nanoparticles in order to increase the intestinal permeability.
- The characteristics and improved intestinal permeability of vancomycin PLGA-nanoparticles as colloidal drug delivery system.
- STUDY OF THE CORRELATION BETWEEN THERMODYNAMIC PARAMETERS AND SOME PHYSICOCHEMICAL AND PHARMACOKINETIC PARAMETERS
- Developments in Methods for Measuring the Intestinal Absorption of Nanoparticle-Bound Drugs
- Crystal-liquid Fugacity Ratio as a Surrogate Parameter for Intestinal Permeability.
- Biowaiver or Bioequivalence: Ambiguity in Sildenafil Citrate BCS Classification
- Bortezomib-loaded solid lipid nanoparticles: preparation, characterization, and intestinal permeability investigation
- Integrating theoretical and experimental permeability estimations for provisional biopharmaceutical classification: Application to the WHO essential medicines
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