An exact mathematical expression for describing competitive binding of two different ligands to a protein molecule

Keywords

Dissociation constant, Expression (computer science), Competitive binding, Constant (computer programming), Dissociation (chemistry)

References

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• A Fluorescence Anisotropy–Based Myt1 Kinase Binding AssayAlexander Rohe, Claudia Henze, Frank Erdmann — 2014
• Nuclear Localization of the DNA Repair Scaffold XRCC1: Uncovering the Functional Role of a Bipartite NLSThomas W. Kirby, Natalie R. Gassman, Cassandra Smith — 2015
• Protein-ligand interactions: fundamentals.Mark A. Williams — 2013
• The Auto-inhibitory Function of Importin α Is Essentialin Vivo *Michelle T. Harreman, Mary R. Hodel, Patrizia Fanara — 2003
• Self-assembly and catalytic activity of the pyruvate dehydrogenase multienzyme complex from Bacillus stearothermophilus.Gonzalo J. Domingo, Hitesh J. Chauhan, Ivan A.D. Lessard — 1999
• Dissecting the nucleotide binding properties of Escherichia coli 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase with fluorescent 3'(2)'-o-anthraniloyladenosine 5'-triphosphate.Genbin Shi, Yunchen Gong, Alexei Savchenko — 2000
• Measurement of dissociation constants of inhibitors binding to Src SH2 domain protein by non‐covalent electrospray ionization mass spectrometryS. W. Annie Bligh, Terry Haley, Peter N. Lowe — 2003
• In vitro influence of fatty acids and bilirubin on binding of mycophenolic acid to human serum albumin.Yoann Vial, Michel Tod, Marilyne Hornecker — 2011
• Biophysical and biochemical analysis of hnRNP K: arginine methylation, reversible aggregation and combinatorial binding to nucleic acidsBodo Moritz, Hauke Lilie, Isabel S. Naarmann‐de Vries — 2014
• Budded baculoviruses as a tool for a homogeneous fluorescence anisotropy-based assay of ligand binding to G protein-coupled receptors: the case of melanocortin 4 receptors.Santa Veikšina, Sergei Kopanchuk, Ago Rinken — 2014
• Analytical expressions for the homotropic binding of ligand to protein dimers and trimersScott T. Lefurgy, Thomas S. Leyh — 2011
• A fluorescence polarization-based assay for peptidyl prolyl cis/trans isomerase cyclophilin A.Yaya Liu, Jianjun Jiang, Paul L. Richardson — 2006
• High-affinity bisubstrate probe for fluorescence anisotropy binding/displacement assays with protein kinases PKA and ROCK.Angela Vaasa, Indrek Viil, Erki Enkvist — 2009
• Identification and functional characterization of a novel acetylcholine-binding protein from the marine annelid Capitella teleta.Thomas McCormack, Robert M. Petrovich, Kelly Mercier — 2010
• Competitive displacement of cofilin can promote actin filament severingW. Austin Elam, Hyeran Kang, Enrique M. De La Cruz — 2013

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