Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions.
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- Type
- article
- Published
- 2007-03-19
- Cited by
- 123
- References
- 36
- Access
- Open access
- OpenAlex
- https://openalex.org/W1966889781
- Semantic Scholar
- https://api.semanticscholar.org/CorpusID:11555546
Keywords
Indole test, Catalysis, Chemistry, Domino, Copper
References
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- Villagorgin A and B. New type of indole alkaloids with acetylcholine antagonist activity from the gorgonian Villagorgia rubra
- On inventing reactions for atom economy.
- Calindol, a Positive Allosteric Modulator of the Human Ca2+ Receptor, Activates an Extracellular Ligand-binding Domain-deleted Rhodopsin-like Seven-transmembrane Structure in the Absence of Ca2+*
- Palladium(0)-catalyzed tandem cyclization of allenenes: direct construction of tricyclic heterocycles through aromatic C--H activation.
- 2-Aryl and 2-heteroaryl indoles from 1-alkynes and o-iodotrifluoroacetanilide through a domino copper-catalyzed coupling-cyclization process.
- Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: diastereoselective access to bicyclic nitrogen heterocycles.
- Molecular determinants of MAO selectivity in a series of indolylmethylamine derivatives: biological activities, 3D-QSAR/CoMFA analysis, and computational simulation of ligand recognition.
- Synthesis and functionalization of indoles through palladium-catalyzed reactions.
- Three-dimensional quantitative structure-activity relationship studies on selected MT1 and MT2 melatonin receptor ligands: requirements for subtype selectivity and intrinsic activity modulation.
- Three-component indole synthesis using ortho-dihaloarenes
- Dopamine D4 ligands and models of receptor activation: 2-(4-pyridin-2-ylpiperazin-1-ylmethyl)-1H-benzimidazole and related heteroarylmethylarylpiperazines exhibit a substituent effect responsible for additional efficacy tuning.
- Observation on the synthesis of allenes by homologation of alk-1-ynes
- Efficient access to azaindoles and indoles.
- Binding of beta-carbolines at imidazoline I2 receptors: a structure-affinity investigation.
- A practical mild, one-pot, regiospecific synthesis of 2,3-disubstituted indoles via consecutive Sonogashira and Cacchi reactions.
- Palladium-catalyzed synthesis of 2-(aminomethyl)indoles from ethyl 3-(o-trifluoroacetamidophenyl)-1-propargyl carbonate.
- A further study of the cytotoxic constituents of a milnamide-producing sponge.
- N2-benzyl-N1-(1-(1-naphthyl)ethyl)-3-phenylpropane-1,2-diamines and conformationally restrained indole analogues: development of calindol as a new calcimimetic acting at the calcium sensing receptor.
- Practical methodologies for the synthesis of indoles.
Cited by
- Synthesis of iodo-indoloazepinones in an iodine-mediated three-component domino reaction via a regioselective 7-endo-dig iodo-cyclization pathway.
- Reductive Alkylation of α-Keto Imines Catalyzed by PTSA/FeCl3: Synthesis of Indoles and 2,3'-Biindoles.
- Carbohydrates as a reagent in multicomponent reactions: one-pot access to a new library of hydrophilic substituted pyrimidine-fused heterocycles.
- Regio- and stereoselective synthesis of a library of bioactive dispiro-oxindolo/acenaphthoquino andrographolides via 1,3-dipolar cycloaddition reaction under microwave irradiation.
- A New Multicomponent Reaction Catalyzed by a Lewis Acid Catalyst: Convenient Synthesis of Polyfunctional Tetrahydropyrimidines
- Electrochemical-Mediated Cyclization of 2-Alkynylanilines: A Clean and Safe Synthesis of Indole Derivatives
- Iridium(III) Cp* Complexes for the Efficient Hydroamination of Internal Alkynes
- A walk around the A3-coupling.
- PPh3-catalyzed synthesis of multifunctional vinylesters from terminal alkynoates and aromatic aldehydes
- Ultrasound-promoted regioselective and stereoselective synthesis of novel spiroindanedionepyrrolizidines by multicomponent 1,3-dipolar cycloaddition of azomethine ylides
- A one-pot three-component reaction involving 2-aminochromone in aqueous micellar medium: a green synthesis of hexahydrochromeno[2,3-bb]quinolinedione
- Recent advances in the synthesis of indole and quinoline derivatives through cascade reactions.
- Ytterbium Triflate Promoted One-Pot Three Component Synthesis of 3,4,5-Trisubstituted-3,6-dihydro-2H-1,3-oxazines
- Sulfur‐Assisted and 1,8‐Diazabicyclo[5.4.0]undec‐7‐ene (DBU)‐Catalyzed Cyclization of 2‐Alkynylanilines for the Metal‐Free Synthesis of Indole Derivatives
- A First Resource-Efficient and Highly Flexible Procedure for a Four-Component Synthesis of Dispiropyrrolidines
- First Synthesis of α,β‐Unsaturated Lactones with High Diversity through the Passerini Reaction and Ring‐Closing Metathesis (RCM)
- Gold(III) stabilized over ionic liquids grafted on MCM-41 for highly efficient three-component coupling reactions.
- Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation.
- Copper catalysis in the construction of indole and benzo[b]furan rings.
- One-pot synthesis of substituted indoles via titanium(IV) alkoxide mediated imine formation – copper-catalyzed N-arylation
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