Inhibition of G protein-coupled receptor signaling by expression of cytoplasmic domains of the receptor.
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Summary
The present studies performed to test the generality as well as the specificity of 3i domain-induced inhibition of receptor activity and suggest that peptides derived from a G protein-coupled receptor might serve as antagonists of receptor/G protein interactions.
- Type
- article
- Published
- 1994-06-03
- Cited by
- 91
- References
- 0
- Access
- Open access
- OpenAlex
- https://openalex.org/W161360456
- Semantic Scholar
- https://api.semanticscholar.org/CorpusID:40937036
Keywords
Cell biology, Receptor, 5-HT5A receptor, Cytoplasm, Signal transduction
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